Drugbank Info

Gene Info

  • Species: Human (Homo sapiens)
  • GeneID: 23621
  • Symbol: BACE1
  • Description: beta-secretase 1
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Drug ID pharmacological_action actions Name Groupo
DB02378 unknown NA MMI-175 experimental
DB06073 yes inhibitor CTS-21166 investigational
DB06930 unknown NA N-[amino(imino)methyl]-2-(2,5-diphenyl-1H-pyrrol-1-yl)acetamide experimental
DB07019 unknown NA N-[(5R,14R)-5-AMINO-5,14-DIMETHYL-4-OXO-3-OXA-18-AZATRICYCLO[15.3.1.1~7,11~]DOCOSA-1(21),7(22),8,10,17,19-HEXAEN-19-YL]-N-METHYLMETHANESULFONAMIDE experimental
DB07089 unknown NA N-[amino(imino)methyl]-2-[2-(2-chlorophenyl)-4-(4-propoxyphenyl)-3-thienyl]acetamide experimental
DB07110 unknown NA 4-(4-FLUOROBENZYL)PIPERIDINE experimental
DB07175 unknown NA N-{2-methyl-5-[(6-phenylpyrimidin-4-yl)amino]phenyl}methanesulfonamide experimental
DB07206 unknown NA 6-[2-(1H-INDOL-6-YL)ETHYL]PYRIDIN-2-AMINE experimental
DB07245 unknown NA 6-[2-(3'-METHOXYBIPHENYL-3-YL)ETHYL]PYRIDIN-2-AMINE experimental
DB07281 unknown NA N~3~-BENZYLPYRIDINE-2,3-DIAMINE experimental
DB07284 unknown NA N~3~-(3-PYRIDIN-3-YLBENZYL)PYRIDINE-2,3-DIAMINE experimental
DB07303 unknown NA N~3~-[3-(5-METHOXYPYRIDIN-3-YL)BENZYL]PYRIDINE-2,3-DIAMINE experimental
DB07345 unknown NA 4-(2-aminoethyl)-2-cyclohexylphenol experimental
DB07346 unknown NA 4-(2-aminoethyl)-2-ethylphenol experimental
DB07415 unknown NA 4-[(1S)-1-(3-fluoro-4-methoxyphenyl)-2-(2-methoxy-5-nitrophenyl)ethyl]-1H-imidazol-2-amine experimental
DB07519 unknown NA (6R)-2-amino-6-[2-(3'-methoxybiphenyl-3-yl)ethyl]-3,6-dimethyl-5,6-dihydropyrimidin-4(3H)-one experimental
DB07535 unknown NA 2-amino-6-[2-(1H-indol-6-yl)ethyl]pyrimidin-4(3H)-one experimental
DB07573 unknown NA (2S)-1-(2,5-dimethylphenoxy)-3-morpholin-4-ylpropan-2-ol experimental
DB07734 unknown NA N-(1-benzylpiperidin-4-yl)-4-sulfanylbutanamide experimental
DB07735 unknown NA N-[1-(2,6-dimethoxybenzyl)piperidin-4-yl]-4-sulfanylbutanamide experimental
DB07736 unknown NA (2S)-4-(4-fluorobenzyl)-N-(2-sulfanylethyl)piperazine-2-carboxamide experimental
DB07737 unknown NA (2S)-4-(4-fluorobenzyl)-N-(3-sulfanylpropyl)piperazine-2-carboxamide experimental
DB07738 unknown NA N-[1-(5-bromo-2,3-dimethoxybenzyl)piperidin-4-yl]-4-sulfanylbutanamide experimental
DB07874 unknown NA (6S)-2-amino-6-(3'-methoxybiphenyl-3-yl)-3,6-dimethyl-5,6-dihydropyrimidin-4(3H)-one experimental
DB07993 unknown NA N~3~-[3-(1H-INDOL-6-YL)BENZYL]PYRIDINE-2,3-DIAMINE experimental
DB07994 unknown NA N~3~-[5-(1H-INDOL-6-YL)-2-(PYRIDIN-2-YLMETHOXY)BENZYL]PYRIDINE-2,3-DIAMINE experimental
DB08749 unknown NA 3-(2-AMINO-6-BENZOYLQUINAZOLIN-3(4H)-YL)-N-CYCLOHEXYL-N-METHYLPROPANAMIDE experimental
DB12285 yes inhibitor Verubecestat investigational