Drugbank Info

Gene Info

  • Species: Human (Homo sapiens)
  • GeneID: 3791
  • Symbol: KDR
  • Description: kinase insert domain receptor
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Drug ID pharmacological_action actions Name Groupo
DB00398 yes antagonist Sorafenib approved|investigational
DB01268 yes inhibitor Sunitinib approved|investigational
DB04727 unknown NA N-(4-{4-AMINO-6-[4-(METHYLOXY)PHENYL]FURO[2,3-D]PYRIMIDIN-5-YL}PHENYL)-N'-[2-FLUORO-5-(TRIFLUOROMETHYL)PHENYL]UREA experimental
DB04849 unknown NA Cediranib investigational
DB04879 unknown NA Vatalanib investigational
DB05014 unknown NA XL999 investigational
DB05075 unknown NA TG-100801 investigational
DB05146 unknown NA XL820 investigational
DB05198 unknown NA CYC116 investigational
DB05578 yes antagonist Ramucirumab approved|investigational
DB06080 unknown NA ABT-869 investigational
DB06101 unknown NA IMC-1C11 investigational
DB06436 unknown NA Semaxanib investigational
DB06589 yes inhibitor Pazopanib approved
DB06595 yes inhibitor Midostaurin approved
DB06626 yes inhibitor Axitinib approved|investigational
DB06938 unknown NA 4-[[2-[[4-chloro-3-(trifluoromethyl)phenyl]amino]-3H-benzimidazol-5-yl]oxy]-N-methyl-pyridine-2-carboxamide experimental
DB07183 unknown NA N-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]nicotinamide experimental
DB07274 unknown NA N-cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide experimental
DB07326 unknown NA 6-chloro-N-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamide experimental
DB07333 unknown NA N-(CYCLOPROPYLMETHYL)-4-(METHYLOXY)-3-({5-[3-(3-PYRIDINYL)PHENYL]-1,3-OXAZOL-2-YL}AMINO)BENZENESULFONAMIDE experimental
DB07334 unknown NA N-[5-(ETHYLSULFONYL)-2-METHOXYPHENYL]-5-[3-(2-PYRIDINYL)PHENYL]-1,3-OXAZOL-2-AMINE experimental
DB07514 unknown NA 3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1H)-one experimental
DB07528 unknown NA 3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1H)-one experimental
DB07537 unknown NA N'-(6-aminopyridin-3-yl)-N-(2-cyclopentylethyl)-4-methyl-benzene-1,3-dicarboxamide experimental
DB08042 unknown NA N~4~-methyl-N~4~-(3-methyl-1H-indazol-6-yl)-N~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine experimental
DB08519 unknown NA N~4~-(3-methyl-1H-indazol-6-yl)-N~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine experimental
DB08875 yes antagonist Cabozantinib approved
DB08896 yes inhibitor Regorafenib approved
DB08901 unknown inhibitor Ponatinib approved
DB09078 yes Inhibitor Lenvatinib approved
DB09079 yes Inhibitor Nintedanib approved
DB12307 unknown NA Foretinib investigational