Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:148
  • Symbol:ADRA1A
  • Description:adrenoceptor alpha 1A
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Drug ID pharmacological_action actions Name Groupo
DB00182 unknown agonist Amphetamine approved|illicit
DB00211 yes agonist Midodrine approved
DB00215 unknown binder Citalopram approved
DB00246 no antagonist Ziprasidone approved
DB00248 unknown binder Cabergoline approved
DB00298 yes antagonist Dapiprazole approved
DB00321 no antagonist Amitriptyline approved
DB00334 unknown antagonist Olanzapine approved|investigational
DB00346 yes antagonist Alfuzosin approved|investigational
DB00363 no antagonist Clozapine approved
DB00368 yes agonist Norepinephrine approved
DB00370 unknown binder Mirtazapine approved
DB00388 yes NA Phenylephrine approved
DB00397 yes agonist Phenylpropanolamine approved|vet_approved|withdrawn
DB00408 unknown binder Loxapine approved
DB00420 unknown antagonist Promazine approved|vet_approved
DB00449 yes agonist Dipivefrin approved
DB00450 yes antagonist Droperidol approved|vet_approved
DB00457 yes antagonist Prazosin approved
DB00458 no antagonist Imipramine approved
DB00477 yes antagonist Chlorpromazine approved|vet_approved
DB00477 unknown NA Chlorpromazine approved|vet_approved
DB00540 no antagonist Nortriptyline approved
DB00543 unknown antagonist Amoxapine approved
DB00543 unknown antagonist Amoxapine approved
DB00575 unknown agonist Clonidine approved
DB00590 yes antagonist Doxazosin approved
DB00598 yes antagonist Labetalol approved
DB00610 yes agonist Metaraminol approved|investigational
DB00622 unknown antagonist Nicardipine approved
DB00656 no antagonist Trazodone approved|investigational
DB00668 yes agonist Epinephrine approved|vet_approved
DB00679 yes antagonist Thioridazine withdrawn
DB00692 yes antagonist Phentolamine approved
DB00696 yes partial agonist Ergotamine approved
DB00699 yes antagonist Nicergoline approved
DB00706 yes antagonist Tamsulosin approved|investigational
DB00723 yes agonist Methoxamine approved
DB00726 unknown antagonist Trimipramine approved
DB00734 unknown antagonist Risperidone approved|investigational
DB00751 unknown unknown Epinastine approved|investigational
DB00777 unknown antagonist Propiomazine approved
DB00797 yes antagonist Tolazoline approved|vet_approved
DB00800 unknown NA Fenoldopam approved
DB00831 yes antagonist Trifluoperazine approved
DB00852 yes agonist Pseudoephedrine approved
DB00865 yes agonist Benzphetamine approved|illicit
DB00875 yes antagonist Flupentixol approved|withdrawn
DB00925 yes antagonist Phenoxybenzamine approved
DB00934 no antagonist Maprotiline approved
DB00935 yes agonist Oxymetazoline approved
DB00964 yes agonist Apraclonidine approved
DB01049 unknown antagonist Ergoloid mesylate approved
DB01069 unknown unknown Promethazine approved
DB01136 yes antagonist Carvedilol approved|investigational
DB01142 unknown antagonist Doxepin approved
DB01149 no antagonist Nefazodone approved|withdrawn
DB01151 no antagonist Desipramine approved
DB01162 yes antagonist Terazosin approved
DB01175 unknown antagonist Escitalopram approved|investigational
DB01186 unknown agonist Pergolide approved|vet_approved|withdrawn
DB01200 unknown agonist Bromocriptine approved|investigational
DB01224 unknown antagonist Quetiapine approved
DB01238 no partial agonist Aripiprazole approved|investigational
DB01253 yes agonist Ergonovine approved
DB01267 unknown antagonist Paliperidone approved
DB01295 unknown antagonist Bevantolol approved
DB01364 unknown inhibitor Ephedrine approved
DB01365 yes agonist Mephentermine approved
DB01403 unknown antagonist Methotrimeprazine approved
DB01472 yes agonist 4-Methoxyamphetamine experimental|illicit
DB01576 unknown antagonist Dextroamphetamine approved|illicit
DB01579 yes agonist Phendimetrazine approved|illicit
DB01614 unknown antagonist Acepromazine approved|vet_approved
DB01622 yes antagonist Thioproperazine approved
DB01624 unknown antagonist Zuclopenthixol approved|investigational
DB04855 unknown antagonist Dronedarone approved
DB04946 unknown antagonist Iloperidone approved
DB05469 unknown NA R450 investigational
DB05492 unknown NA Epicept NP-1 investigational
DB06144 unknown NA Sertindole approved|withdrawn
DB06148 unknown antagonist Mianserin approved
DB06207 yes antagonist Silodosin approved
DB06216 unknown antagonist Asenapine approved
DB06262 yes agonist Droxidopa approved|investigational
DB06694 yes agonist Xylometazoline approved
DB06706 yes agonist Isometheptene approved
DB06711 yes agonist Naphazoline approved
DB06764 yes agonist Tetryzoline approved
DB08922 unknown antagonist Perospirone approved
DB09167 yes inhibitor Dosulepin approved
DB09202 yes agonist Cirazoline experimental