Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:3269
  • Symbol:HRH1
  • Description:histamine receptor H1
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Drug ID pharmacological_action actions Name Groupo
DB00215 unknown binder Citalopram approved
DB00245 unknown antagonist Benzatropine approved
DB00246 no antagonist Ziprasidone approved
DB00283 yes antagonist Clemastine approved
DB00321 no antagonist Amitriptyline approved
DB00334 unknown antagonist Olanzapine approved|investigational
DB00341 yes antagonist Cetirizine approved
DB00342 yes antagonist Terfenadine withdrawn
DB00354 yes antagonist Buclizine approved
DB00363 no antagonist Clozapine approved
DB00366 yes antagonist Doxylamine approved|vet_approved
DB00370 no antagonist Mirtazapine approved
DB00405 yes antagonist Dexbrompheniramine approved
DB00408 unknown binder Loxapine approved
DB00420 unknown antagonist Promazine approved|vet_approved
DB00427 yes antagonist Triprolidine approved
DB00434 yes antagonist Cyproheptadine approved
DB00455 yes antagonist Loratadine approved
DB00458 no antagonist Imipramine approved
DB00477 yes antagonist Chlorpromazine approved|vet_approved
DB00540 no antagonist Nortriptyline approved
DB00543 unknown antagonist Amoxapine approved
DB00557 yes antagonist Hydroxyzine approved
DB00568 yes antagonist Cinnarizine approved
DB00637 yes antagonist Astemizole approved|withdrawn
DB00656 unknown antagonist Trazodone approved|investigational
DB00719 yes antagonist Azatadine approved
DB00726 unknown antagonist Trimipramine approved
DB00734 unknown antagonist Risperidone approved|investigational
DB00737 yes antagonist Meclizine approved
DB00748 yes antagonist Carbinoxamine approved
DB00751 yes antagonist Epinastine approved|investigational
DB00767 yes antagonist Benzquinamide withdrawn
DB00768 yes antagonist Olopatadine approved
DB00777 yes antagonist Propiomazine approved
DB00792 yes antagonist Tripelennamine approved|vet_approved
DB00797 unknown agonist Tolazoline approved|vet_approved
DB00835 yes antagonist Brompheniramine approved
DB00902 yes antagonist Methdilazine approved
DB00920 yes antagonist Ketotifen approved
DB00934 no antagonist Maprotiline approved
DB00950 yes antagonist Fexofenadine approved
DB00967 yes antagonist Desloratadine approved|investigational
DB00972 yes antagonist Azelastine approved
DB00985 yes antagonist Dimenhydrinate approved
DB01069 yes antagonist Promethazine approved
DB01071 yes antagonist Mequitazine approved
DB01075 yes antagonist Diphenhydramine approved
DB01084 yes antagonist Emedastine approved
DB01106 yes antagonist Levocabastine approved
DB01114 yes antagonist Chlorphenamine approved
DB01142 yes antagonist Doxepin approved
DB01146 yes antagonist Diphenylpyraline approved
DB01151 no antagonist Desipramine approved
DB01173 yes antagonist Orphenadrine approved
DB01175 unknown antagonist Escitalopram approved|investigational
DB01176 yes antagonist Cyclizine approved
DB01224 unknown antagonist Quetiapine approved
DB01237 yes antagonist Bromodiphenhydramine approved
DB01238 no antagonist Aripiprazole approved|investigational
DB01239 unknown antagonist Chlorprothixene approved|withdrawn
DB01246 yes antagonist Alimemazine approved|vet_approved
DB01267 unknown agonist Paliperidone approved
DB01403 unknown antagonist Methotrimeprazine approved
DB01615 yes antagonist Aceprometazine approved
DB01619 yes antagonist Phenindamine approved
DB01620 yes antagonist Pheniramine approved
DB01624 unknown antagonist Zuclopenthixol approved|investigational
DB04837 yes antagonist Clofedanol approved|withdrawn
DB04841 unknown antagonist Flunarizine approved
DB04890 yes antagonist Bepotastine approved
DB04905 unknown antagonist Tesmilifene investigational
DB04946 unknown antagonist Iloperidone approved
DB05079 unknown NA HY10275 investigational
DB05080 unknown NA OBE101 investigational
DB05345 unknown NA SO-101 investigational
DB05381 yes agonist Histamine approved|investigational
DB05492 unknown NA Epicept NP-1 investigational
DB06016 yes partial agonist Cariprazine approved
DB06148 unknown antagonist Mianserin approved
DB06216 unknown antagonist Asenapine approved
DB06282 yes antagonist Levocetirizine approved
DB06678 unknown inverse agonist Esmirtazapine investigational
DB06691 yes antagonist Mepyramine approved|vet_approved
DB06698 yes agonist Betahistine approved
DB06766 unknown antagonist Alcaftadine approved
DB08799 yes antagonist Antazoline approved
DB08800 yes antagonist Chloropyramine approved
DB08801 yes antagonist Dimetindene approved
DB08802 yes antagonist Isothipendyl approved
DB08922 unknown inverse agonist Perospirone approved
DB08936 yes antagonist Chlorcyclizine approved
DB09016 yes Inhibitor Butriptyline approved
DB09167 yes antagonist Dosulepin approved
DB09488 yes antagonist Acrivastine approved
DB09555 yes antagonist Dexchlorpheniramine maleate approved
DB11591 yes antagonist Bilastine approved
DB11614 yes antagonist Rupatadine approved