Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:3356
  • Symbol:HTR2A
  • Description:5-hydroxytryptamine receptor 2A
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Drug ID pharmacological_action actions Name Groupo
DB00246 yes antagonist Ziprasidone approved
DB00247 yes antagonist Methysergide approved
DB00248 unknown agonist Cabergoline approved
DB00268 unknown agonist Ropinirole approved|investigational
DB00321 yes antagonist Amitriptyline approved
DB00334 yes antagonist Olanzapine approved|investigational
DB00363 yes antagonist Clozapine approved
DB00370 yes antagonist Mirtazapine approved
DB00408 yes antagonist Loxapine approved
DB00409 unknown other/unknown Remoxipride approved|withdrawn
DB00413 unknown unknown Pramipexole approved|investigational
DB00420 unknown antagonist Promazine approved|vet_approved
DB00434 yes antagonist Cyproheptadine approved
DB00458 unknown antagonist Imipramine approved
DB00477 yes antagonist Chlorpromazine approved|vet_approved
DB00477 unknown NA Chlorpromazine approved|vet_approved
DB00502 unknown other/unknown Haloperidol approved
DB00540 yes antagonist Nortriptyline approved
DB00543 unknown antagonist Amoxapine approved
DB00589 yes agonist Lisuride approved
DB00604 yes agonist Cisapride approved|investigational|withdrawn
DB00656 yes antagonist Trazodone approved|investigational
DB00679 yes antagonist Thioridazine withdrawn
DB00696 yes agonist Ergotamine approved
DB00714 unknown agonist Apomorphine approved|investigational
DB00715 unknown other/unknown Paroxetine approved|investigational
DB00726 unknown agonist Trimipramine approved
DB00734 yes antagonist Risperidone approved|investigational
DB00751 unknown antagonist Epinastine approved|investigational
DB00777 unknown antagonist Propiomazine approved
DB00805 yes antagonist Minaprine approved
DB00843 unknown other/unknown Donepezil approved
DB00875 yes antagonist Flupentixol approved|withdrawn
DB00924 yes antagonist Cyclobenzaprine approved
DB00933 yes antagonist Mesoridazine approved
DB00934 unknown antagonist Maprotiline approved
DB01069 unknown antagonist Promethazine approved
DB01079 unknown antagonist Tegaserod investigational|withdrawn
DB01142 yes antagonist Doxepin approved
DB01149 yes antagonist Nefazodone approved|withdrawn
DB01151 yes antagonist Desipramine approved
DB01186 unknown agonist Pergolide approved|vet_approved|withdrawn
DB01200 unknown agonist Bromocriptine approved|investigational
DB01224 yes antagonist Quetiapine approved
DB01238 yes antagonist Aripiprazole approved|investigational
DB01239 yes antagonist Chlorprothixene approved|withdrawn
DB01242 yes antagonist Clomipramine approved|vet_approved
DB01267 yes antagonist Paliperidone approved
DB01392 unknown antagonist Yohimbine approved|vet_approved
DB01403 unknown antagonist Methotrimeprazine approved
DB01442 yes agonist MMDA experimental|illicit
DB01454 unknown agonist 3,4-Methylenedioxymethamphetamine experimental|illicit
DB01488 unknown NA Dimethyltryptamine experimental|illicit
DB01614 yes antagonist Acepromazine approved|vet_approved
DB01618 unknown antagonist Molindone approved
DB01621 yes antagonist Pipotiazine approved
DB01622 yes antagonist Thioproperazine approved
DB01623 yes antagonist Thiothixene approved
DB01624 unknown antagonist Zuclopenthixol approved|investigational
DB04599 unknown NA Aniracetam experimental
DB04842 unknown antagonist Fluspirilene approved
DB04908 yes antagonist Flibanserin approved
DB04946 yes antagonist Iloperidone approved
DB05079 unknown NA HY10275 investigational
DB05227 unknown NA APD791 investigational
DB05316 yes inverse agonist Pimavanserin investigational
DB05492 unknown NA Epicept NP-1 investigational
DB05687 unknown NA BL-1020 investigational
DB06016 yes agonist Cariprazine approved
DB06077 unknown NA Lumateperone investigational
DB06144 yes antagonist Sertindole approved|withdrawn
DB06148 unknown antagonist Mianserin approved
DB06216 yes antagonist Asenapine approved
DB06288 unknown antagonist Amisulpride approved|investigational
DB06512 unknown antagonist Deramciclane investigational
DB06678 unknown inverse agonist Esmirtazapine investigational
DB08810 yes antagonist Cinitapride approved
DB08815 yes antagonist Lurasidone approved
DB08922 yes inverse agonist Perospirone approved
DB08927 unknown antagonist Amperozide experimental
DB09016 yes antagonist Butriptyline approved
DB09128 yes agonist Brexpiprazole approved
DB09167 yes antagonist Dosulepin approved
DB12555 unknown NA Nelotanserin investigational