Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:5604
  • Symbol:MAP2K1
  • Description:mitogen-activated protein kinase kinase 1
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Drug ID pharmacological_action actions Name Groupo
DB02152 unknown NA K-252a experimental
DB03115 unknown NA 5-Bromo-N-(2,3-Dihydroxypropoxy)-3,4-Difluoro-2-[(2-Fluoro-4-Iodophenyl)Amino]Benzamide experimental
DB05239 yes inhibitor Cobimetinib approved
DB06616 unknown inhibitor Bosutinib approved
DB06892 unknown NA (5S)-4,5-difluoro-6-[(2-fluoro-4-iodophenyl)imino]-N-(2-hydroxyethoxy)cyclohexa-1,3-diene-1-carboxamide experimental
DB07046 unknown NA 2-[(2-chloro-4-iodophenyl)amino]-N-{[(2R)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamide experimental
DB07101 unknown NA PD-0325901 investigational
DB08130 unknown NA N-(5-{3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]phenyl}-1,3,4-oxadiazol-2-yl)ethane-1,2-diamine experimental
DB08208 unknown NA 2-[(4-ETHYNYL-2-FLUOROPHENYL)AMINO]-3,4-DIFLUORO-N-(2-HYDROXYETHOXY)BENZAMIDE experimental
DB08911 yes inhibitor Trametinib approved