Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:4986
  • Symbol:OPRK1
  • Description:opioid receptor kappa 1
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Drug ID pharmacological_action actions Name Groupo
DB00193 unknown agonist Tramadol approved|investigational
DB00295 yes agonist Morphine approved|investigational
DB00318 yes partial agonist Codeine approved|illicit
DB00321 unknown agonist Amitriptyline approved
DB00327 yes agonist Hydromorphone approved|illicit
DB00370 unknown agonist Mirtazapine approved
DB00396 unknown activator Progesterone approved|vet_approved
DB00454 yes antagonist Pethidine approved
DB00497 yes agonist Oxycodone approved|illicit|investigational
DB00514 unknown agonist Dextromethorphan approved
DB00611 yes agonist Butorphanol approved|illicit|vet_approved
DB00647 yes antagonist Dextropropoxyphene approved|illicit|withdrawn
DB00652 yes agonist Pentazocine approved|vet_approved
DB00704 yes antagonist Naltrexone approved|investigational|vet_approved
DB00708 unknown other Sufentanil approved|investigational
DB00813 unknown agonist Fentanyl approved|illicit|investigational|vet_approved
DB00825 unknown agonist Menthol approved
DB00836 yes agonist Loperamide approved
DB00844 yes agonist Nalbuphine approved
DB00854 unknown agonist Levorphanol approved
DB00899 unknown agonist Remifentanil approved
DB00921 yes antagonist Buprenorphine approved|illicit|investigational|vet_approved
DB01183 yes antagonist Naloxone approved|vet_approved
DB01209 yes antagonist Dezocine approved
DB01221 unknown agonist Ketamine approved|vet_approved
DB01439 yes agonist 3-Methylthiofentanyl experimental|illicit
DB01452 unknown agonist Heroin approved|illicit
DB01497 yes agonist Etorphine illicit|vet_approved
DB01535 unknown agonist Carfentanil illicit|vet_approved
DB01548 unknown antagonist Diprenorphine illicit|vet_approved
DB01565 unknown agonist Dihydromorphine experimental|illicit
DB01571 yes agonist 3-Methylfentanyl illicit
DB05046 unknown NA V1003 investigational
DB05104 unknown NA Asimadoline investigational
DB05155 unknown NA CR665 investigational
DB05443 unknown NA ADL 10-0101 investigational
DB06148 unknown agonist Mianserin approved
DB06204 unknown inhibitor Tapentadol approved
DB06274 unknown antagonist Alvimopan approved
DB06738 yes agonist Ketobemidone approved
DB06800 no antagonist Methylnaltrexone approved
DB09272 yes agonist Eluxadoline approved
DB09396 yes agonist Propoxyphene napsylate approved