Drugbank Info

Gene Info

  • Species:Human (Homo sapiens)
  • GeneID:4988
  • Symbol:OPRM1
  • Description:opioid receptor mu 1
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Drug ID pharmacological_action actions Name Groupo
DB00193 yes agonist Tramadol approved|investigational
DB00295 yes agonist Morphine approved|investigational
DB00318 yes partial agonist Codeine approved|illicit
DB00321 unknown binder Amitriptyline approved
DB00327 yes agonist Hydromorphone approved|illicit
DB00333 yes agonist Methadone approved
DB00497 yes agonist Oxycodone approved|illicit|investigational
DB00504 yes partial agonist Levallorphan approved
DB00514 unknown agonist Dextromethorphan approved
DB00611 yes partial antagonist Butorphanol approved|illicit|vet_approved
DB00647 yes agonist Dextropropoxyphene approved|illicit|withdrawn
DB00652 yes antagonist Pentazocine approved|vet_approved
DB00704 yes antagonist Naltrexone approved|investigational|vet_approved
DB00708 yes agonist Sufentanil approved|investigational
DB00802 yes agonist Alfentanil approved|illicit
DB00813 yes agonist Fentanyl approved|illicit|investigational|vet_approved
DB00836 yes agonist Loperamide approved
DB00844 yes antagonist Nalbuphine approved
DB00854 yes agonist Levorphanol approved
DB00899 yes agonist Remifentanil approved
DB00904 unknown other/unknown Ondansetron approved
DB00913 yes agonist Anileridine approved|illicit
DB00921 yes partial agonist Buprenorphine approved|illicit|investigational|vet_approved
DB00956 yes agonist Hydrocodone approved|illicit
DB01081 yes agonist Diphenoxylate approved|illicit
DB01183 yes antagonist Naloxone approved|vet_approved
DB01192 yes agonist Oxymorphone approved|investigational|vet_approved
DB01209 yes agonist Dezocine approved
DB01221 unknown binder Ketamine approved|vet_approved
DB01227 yes agonist Levomethadyl Acetate approved
DB01433 yes agonist Methadyl Acetate approved|illicit
DB01439 yes agonist 3-Methylthiofentanyl experimental|illicit
DB01444 yes agonist Dimethylthiambutene experimental|illicit
DB01452 yes agonist Heroin approved|illicit
DB01466 yes agonist Ethylmorphine approved|illicit
DB01497 yes agonist Etorphine illicit|vet_approved
DB01535 yes agonist Carfentanil illicit|vet_approved
DB01548 yes antagonist Diprenorphine illicit|vet_approved
DB01565 yes agonist Dihydromorphine experimental|illicit
DB01571 yes agonist 3-Methylfentanyl illicit
DB05046 unknown NA V1003 investigational
DB05492 unknown NA Epicept NP-1 investigational
DB05509 unknown NA LI-301 investigational
DB06204 yes agonist Tapentadol approved
DB06274 yes antagonist Alvimopan approved
DB06738 yes agonist Ketobemidone approved
DB06800 yes antagonist Methylnaltrexone approved
DB09049 yes antagonist Naloxegol approved
DB09089 yes agonist Trimebutine approved
DB09272 yes agonist Eluxadoline approved
DB09396 yes agonist Propoxyphene napsylate approved